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Template:Relative potencies of selected antiandrogens

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Relative potencies of selected antiandrogens
Antiandrogen Relative potency
Bicalutamide 4.3
Hydroxyflutamide 3.5
Flutamide 3.3
Cyproterone acetate 1.0
Zanoterone 0.4
Description: Relative potencies of orally administered antiandrogens in antagonizing 0.8 to 1.0 mg/kg s.c.Tooltip subcutaneous injection testosterone propionate-induced ventral prostate weight increase in castrated immature male rats. Higher values mean greater potency. Sources: [1]

References

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  1. ^ Snyder BW, Winneker RC, Batzold FH (December 1989). "Endocrine profile of Win 49596 in the rat: a novel androgen receptor antagonist". J. Steroid Biochem. 33 (6): 1127–32. doi:10.1016/0022-4731(89)90419-6. PMID 2615357.